Benzothiazolyl ureas are low micromolar and uncompetitive inhibitors of 17β-HSD10 with implications to Alzheimer’s disease treatment

Schmidt, M., Benek, O., Vinklarova, L., Hrabinova, M., Zemanova, L., Chribek, M., Kralova, V., Hroch, L., Dolezal, R., Lycka, A., Prchal, L., Jun, D., Aitken, L., Gunn-Moore, F., Kuca, K. & Musilek, K., 17 Mar 2020, In: International Journal of Molecular Sciences. 21, 6, 26 p., 2059.

Research output: Contribution to journal › Article › peer-review

Neuroprotective actions of leptin facilitated through balancing mitochondrial morphology and improving mitochondrial function

Cheng, Y., Buchan, M., Vitanova, K., Aitken, L., Gunn-Moore, F. J., Ramsay, R. R. & Doherty, G., 13 Oct 2020, In: Journal of Neurochemistry. 155, 2, p. 191-206 e15003.

Research output: Contribution to journal › Article › peer-review

Tacrine – benzothiazoles: novel class of potential multitarget anti-Alzheimeŕs drugs dealing with cholinergic, amyloid and mitochondrial systems

Nepovimova, E., Svobodova, L., Dolezal, R., Hepnarova, V., Junova, L., Jun, D., Korabecny, J., Kucera, T., Gazova, Z., Motykova, K., Kubackova, J., Bednarikova, Z., Janockova, J., Jesus, C., Cortes, L., Pina, J., Rostohar, D., Serpa, C., Soukup, O., Aitken, L. & 10 others, Hughes, R. E., Musilek, K., Muckova, L., Jost, P., Chvojkova, M., Vales, K., Valis, M., Chrienova, Z., Chalupova, K. & Kuca, K., 28 Dec 2020, In: Bioorganic Chemistry. In-Press, 104596.

Research output: Contribution to journal › Article › peer-review